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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T13016 | SR59230A | Adrenergic Receptor | |
SR59230A is a potent, selective antagonist of β3-adrenergic receptor(β3, β1, and β2 receptors with IC50s of 40, 408, and 648 nM , respectively). | |||
T82407 | Feruloyl tyramine | ||
Feruloyl tyramine, an amide isolated from the ethanol extract of hemp seeds, induces hypothermia and dyskinesia when injected into the lateral ventricle of mice [1]. | |||
T29206 | ZCZ011 | ZCZ 011,ZCZ-011 | |
ZCZ011 is a positive allosteric modulator of the cannabinoid CB1 receptor. ZCZ011 is brain penetrant, increased the potency of orthosteric agonists in mouse behavioral assays indicative of cannabimimetic activity, includ... | |||
T28845 | SR142948A HCl | SR142948A,SR 142948A,SR-142948A,SR142948A hydrochloride | |
SR 142948A is a non-peptide antagonist of neurotensin receptor. SR 142948A affects the expression of c-Fos and has properties of antipsychotic agent. SR 142948A blocks hypothermia and analgesia induced by neurotensin. It... | |||
T38007 | Noladin ether | ||
Noladin ether is a selective cannabinoid CB1 receptor agonist (Ki=21.2 nM). Noladin ether can cause hypothermia, intestinal immobility, and mild pain relief. | |||
T72395 | CB1 inverse agonist 2 | ||
CB1 Inverse Agonist 2, an orally active compound, serves as an inverse agonist for the Cannabinoid Receptor CB1. It effectively counteracts the hypothermia and anorexia induced by CP55940 in mouse models. | |||
T38138 | ACEA | 2'-chloro-AEA,Arachidonoyl 2'-Chloroethylamide | |
Arachidonoyl 2-chloroethylamide (ACEA) is a potent and selective cannabinoid (CB) receptor 1 agonist with Ki values of 1.4 and >2,000 nM for CB1 and CB2 receptors, respectively. In whole animal experiments, ACEA induces ... | |||
T73677 | SR 142948 dihydrochloride | ||
SR 142948 dihydrochloride is a selective, orally active, non-peptide neurotensin receptor (NT) antagonist, featuring IC50 values of 1.19 nM, 0.32 nM, and 3.96 nM in h-NTR1-CHO cells, HT-29 cells, and adult rat brain, res... |