20
Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T40117 | Antileishmanial agent-1 | ||
Antileishmanial agent-1 demonstrates activity against both L. amazonensis promastigotes (IC 50 = 15.52 μM) and intracellular amastigotes (IC 50 = 4.10 μM). | |||
T79449 | Antileishmanial agent-19 | Parasite | |
Compound F27 (Antileishmanial agent-19) is an antileishmanial compound effective against L. donovani promastigotes, demonstrating an IC50 of 3.39 μM. It functions by inhibiting the Leishmania prolyl-tRNA synthetase and d... | |||
T78964 | Antileishmanial agent-17 | Parasite | |
Antileishmanial agent-17, a coumarin hybrid, exhibits potent antileishmanial activity (IC50 <0.78 μM) while proving non-toxic to normal VERO cells. It specifically interacts with the folate pathway enzymes pteridine redu... | |||
T79471 | Antileishmanial agent-20 | Parasite | |
Antileishmanial agent-20 exhibits selectivity against the Leishmania parasite, with IC50 values of 2.8 μM for L. infantum and 0.2 μM for L. braziliensis. It is a potential research tool for studying these parasites [1]. | |||
T60638 | Antileishmanial agent-8 | ||
Antileishmanial agent-8 (compound 18) shows potent and selective activity against Leishmania donovani ( L. donovani ) (IC50 = 5.64 μM) with relatively low cytotoxicity in L-6 cells (IC 50 =73.9 μM) [1]. | |||
T79633 | Antileishmanial agent-22 | Parasite | |
Antileishmanial agent-22 (compound 15b) serves as an antiparasitic and antibacterial, exhibiting activities against Leishmania (IC50 = 0.408 μM), malaria, and tuberculosis. It operates on an antifolate mechanism, suppres... | |||
T61199 | Antileishmanial agent-2 | ||
Antileishmanial agent-2 demonstrates potent submicromolar antileishmanial activity (IC50 = 0.29 μM) and a remarkable selectivity index against mammalian cells. | |||
T61710 | Antileishmanial agent-7 | ||
Antileishmanial agent-7 (compound 23) exhibits strong antileishmanial activity against Leishmania donovani and L-6, with IC50 values of 6.89 and 259 μM, respectively [1]. | |||
T61391 | Antileishmanial agent-3 | ||
Antileishmanial agent-3 (Compound 13) effectively inhibits the growth of Leishmania major [1]. | |||
T63281 | Antileishmanial agent-11 | ||
Antileishmanial agent-11 is a potent antileishmanial agent that acts on Leishmania brazilensis (IC50: 28.3 μM), Leishmania infantum (IC50: 24.8 μM) and T. cruzi (IC50: 13.0 μM) with outstanding antiprotozoal effect. | |||
T62574 | Antileishmanial agent-6 | ||
Antileishmanial agent-6 is a potent anti-leishmanial agent with anti-leishmanial activity (IC50: 0.54 μM) and cytotoxicity (IC50: 10.2 μM) against Leishmania donovani and L-6. | |||
T61560 | Antileishmanial agent-5 | ||
Antileishmanial agent-4 is a ribonucleoside analogue with potent activity against L.infantum and T.cruzi, having EC 50 values of 0.68 μM and 0.83 μM, respectively [1]. | |||
T78963 | Antileishmanial agent-16 | Parasite | |
Antileishmanial agent-16 (compound 14c), an anti-Leishmania agent, exhibits potent activity against Leishmania major promastigotes (IC50 = 0.59 µM) and amastigotes (IC50 = 0.81 µM), while maintaining a favorable safety p... | |||
T61100 | Antileishmanial agent-4 | ||
Antileishmanial agent-4, a ribonucleoside analogue, functions as an antileishmanial agent [1]. | |||
T79419 | Antileishmanial agent-24 | Parasite | |
Antileishmanial agent-24 (compound 33) exhibits antileishmanial activity, demonstrating an inhibitory concentration 50 (IC50) value of 5.39 μM against amastigotes [1]. | |||
T62210 | Antileishmanial agent-10 | ||
Antileishmanial agent-10 (Compound 7h) is an antiprotozoal agent. | |||
T72260 | Antileishmanial agent-13 | ||
Antileishmanial agent-13, a quinoline-isatin hybrid, functions as an antileishmanial agent targeting the L. Major Leishmania strain through an anti-folate mechanism. This compound exhibits potent inhibition of both the p... | |||
T83045 | Antileishmanial agent-25 | Parasite | |
Antileishmanial agent-25 (compound 24) exhibits selective activity against intracellular amastigotes, demonstrating an inhibitory concentration (IC50) of 6.63 μM [1]. | |||
T79632 | Antileishmanial agent-21 | Parasite | |
Antileishmanial agent-21 (compound 4e) functions as an inhibitor of Leishmania pteridine reductase 1 (Lm-PTR1), employing an anti-folate mechanism. Its antileishmanial effects can be negated by folic acid and leucovorin.... | |||
T78680 | Antileishmanial agent-14 | Parasite | |
Antileishmanial agent-14, a sulfuretin analog, exhibits potential activity against Leishmania donovani promastigotes (IC 50 = 4.1 μM) and inhibits infection by L. donovani amastigotes (IC 50 = 11.1 μM) [1]. |