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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T11005 | Desmethyl Celecoxib | COX | |
Demethyl celecoxib is a selective inhibitor of COX-2 with anti-inflammatory activity (IC50 of 32 nM). with anti-inflammatory activities. Desmethyl Celecoxib is an analog of Celecoxib and with the optimal yield of 75%. | |||
T22632 | TASIN-1 | 1-[(4-methoxyphenyl)sulfonyl]-4'-methyl-4,1'-bipiperidine | APC |
TASIN-1 is a small molecule inhibitor of mutant adenomatous polyposis coli (APC). | |||
T81876 | MAIT-203 | ||
MAIT-203, a cyclopentyalanin-derived peptidomimetic, effectively disrupts the interaction between adenomatous polyposis coli (APC) and Asef (RhoGEF4), without affecting APC-Sam68 or APC-striatin interactions. It binds to... | |||
T32026 | GYKI-13324 | GYKI 13324,GYKI13324 | |
GYKI-13324 is bifunctional nitrosoureido derivative and alkylating agent. GYKI-13324 was studied on human colorectal tumor xenograft lines. Given orally in single or multiple daily doses, GYKI-13324 produced long-term or... |