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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T13394 | ZEN-3862 | ZEN3862,ZEN 3862 | Epigenetic Reader Domain |
ZEN-3862 (Willardiine) is an inhibitor of BET(IC50s of 0.16 and 0.13 μM for BRD4(BD1) and BRD4(BD2) , respectively). ZEN-3862 can be used to form PROTACs to induce degradation of BRD4. |