Home Tools
Log in
Cart

Search Result

Search Results for " varenicline "

5

Compounds

Cat No. Product Name Synonyms Targets
T4246L Varenicline
Varenicline (CP 526555), a cytisine-based nicotinic ligand, is a potent partial agonist for the α4β2 nicotinic acetylcholine receptor (nAChR) with an EC50 value of 2.3 μM and acts as a full agonist for α7 and α3β4 nAChRs...
T4246 Varenicline dihydrochloride AChR
Varenicline dihydrochloride is a Selective α4β2 nicotinic acetylcholine receptor partial agonist.
T1657 Varenicline Tartrate Champix tartrate,Chantix tartrate,CP 526555-18 AChR
Varenicline Tartrate (CP 526555-18) is a benzazepine derivative that functions as an ALPHA4/BETA2 NICOTINIC RECEPTOR partial agonist. It is used for SMOKING CESSATION.
T23502 Varenicline Hydrochloride Others
Varenicline Hydrochloride is a partial agonist of α4β2 nicotinic receptor.
T36810 UPSEM 792 hydrochloride
Ultrapotent PSEM (uPSEM) agonist for PSAM4-GlyR and PSAM4-5HT3 (Ki = 0.7 nM for PSAM4-GlyR and <10 nM for PSAM4-5HT3). Exhibits >10,000-fold agonist selectivity for PSAM4-GlyR over α7-GlyR, α7-5HT3, and 5HT3-R, and 230-f...
TargetMol