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Cat No. | Product Name | Synonyms | Targets |
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TP1205 | Velmupressin acetate | V2 receptor (V2R) agonist,c(Bua-Cpa-Thi-Val-Asn-Cys)-Pro-d-Arg-NEt2 acetate | |
c(Bua-Cpa-Thi-Val-Asn-Cys)-Pro-d-Arg-NEt2 acetate is a potent, selective and short-acting peptidic V2 receptor (V2R) agonist with EC50s of 0.07 and 0.02 nM for hV2R and rV2R, respectively. | |||
T15273 | Fedovapagon | VA483,A106483 | Vasopressin Receptor |
Fedovapagon (VA106483) is a selective and potent agonist of the vasopressin V2 receptor (V2R) that inhibits the growth of intersegmental vessels in zebrafish. Fedovapagon can be used to study overactive bladder, nocturia... | |||
TP1560 | C(Bua-Cpa-Thi-Val-Asn-Cys)-Pro-Agm | ||
c(Bua-Cpa-Thi-Val-Asn-Cys)-Pro-Agm a highly efficient, selective and short-acting peptide V2 receptor agonist (V2R), with EC50s of hV2R and rV2R being 0.25 and 0.05 nM, respectively. | |||
T64174 | Vasopressin V2 receptor antagonist 1 | ||
Vasopressin V2 receptor antagonist 1 (Compound 4g) is a vasopressin V2receptor (V2R) antagonist (Ki: 3.8 nM). dominant polycystic kidney disease (ADPKD). | |||
T80198 | Vasopressin Dimer (anti-parallel) (TFA) | Vasopressin Receptor | |
Vasopressin Dimer (anti-parallel) TFA, an anti-parallel dimer form of vasopressin, has the capability to activate four G protein-coupled receptors: V1aR, V1bR, V2R, and OTR [1]. | |||
T80197 | Vasopressin Dimer (parallel) (TFA) | Vasopressin Receptor | |
Vasopressin Dimer (parallel) TFA, a parallel dimer of Vasopressin, has the capability to activate four G protein-coupled receptors—namely, V1aR, V1bR, V2R, and OTR [1]. | |||
TP1473 | Velmupressin | c(Bua-Cpa-Thi-Val-Asn-Cys)-Pro-d-Arg-NEt2 | |
c(Bua-Cpa-Thi-Val-Asn-Cys)-Pro-d-Arg-NEt2 is a selective and short-acting peptidic V2 receptor (V2R) agonist with EC50s of 0.07nM and 0.02 nM for hV2R and rV2R, respectively. | |||
T80138 | (D-Arg8)-Inotocin | Vasopressin Receptor | |
'(D-Arg8)-Inotocin is a potent, selective, and competitive antagonist of the vasopressin receptor (V 1a R), exhibiting a binding affinity (K i) of 1.3 nM. It demonstrates over 3000-fold selectivity for the human V1aR com... |
Cat No. | Product Name | Species | Expression System |
---|---|---|---|
TMPH-03132 | AVPR2 Protein, Pig, Recombinant (His & SUMO) | Sus scrofa (Pig) | E. coli |
Receptor for arginine vasopressin. The activity of this receptor is mediated by G proteins which activate adenylate cyclase. Involved in renal water reabsorption. |