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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T79772 | RARα antagonist 1 | Others | |
Compound 21, an orally active and selective RARα antagonist, exhibits a potent inhibition of the retinoic acid receptor α with an IC50 of 4.6 nM [1]. | |||
T14143 | AGN 194310 | VTP-194310 | Retinoid Receptor |
AGN 194310 (VTP-194310) is retinioic acid receptors (RARs) pan-antagonist. The Kd values of 3 nM, 2 nM, 5 nM for RARα, RARβ, RARγ, respectively[1][2]. | |||
T78102 | ER 50891 quarterhydrate | Others | |
ER 50891 quarterhydrate is a potent RARα (retinoic acid receptor α) antagonist that markedly diminishes the inhibitory effects of ATRA (all-trans retinoic acid) on osteoblastogenesis induced by BMP 2 (bone morphogenetic ... | |||
T85283 | AGN 193109 sodium | CD3106 | Others |
AGN 193109 is a potent antagonist of retinoic acid receptors (RARs; Kd= 2, 2, and 3 nM for RARα, β, and γ, respectively), exhibiting selectivity for RARs over retinoid X receptors (RXRs; Kd= >10,000 nM for human RXRα, β,... |