prmt-1-in-1 — TargetMol Chemicals

Cat No.	Product Name	Synonyms	Targets
T12541	PRMT5-IN-1		Histone Methyltransferase
	PRMT5-IN-1 is a covalent inhibitor of protein arginine methyltransferase 5 (PRMT5)(IC50 of 11 nM for PRMT5/MEP50).		Histone Methyltransferase
T38421	PRMT1-IN-1	PRMT1-IN-1
	PRMT1-IN-1 is a PRMT1 inhibitor.
T4013	SGC2085 HCl		Histone Methyltransferase
	SGC2085 is a potent and selective coactivator associated arginine methyltransferase 1 (CARM1) Inhibitor with an IC50 of 50 nM and more than undred-fold selectivity over other PRMTs. CARM1 is an important positive modulat...		Histone Methyltransferase
T81399	PRMT4-IN-2
	PRMT4-IN-2 (compound 55) acts as a pan-inhibitor across various protein arginine methyltransferase (PRMT) isoforms, exhibiting inhibitory potencies with IC50 values of 92 nM for PRMT4, 436 nM for PRMT6, 460 nM for PRMT1,...
T79355	PRMT4-IN-3		Histone Methyltransferase
	PRMT4-IN-3 (compound 56) serves as a potent class I protein arginine methyltransferase (PRMT) inhibitor, specifically targeting PRMT4 with an IC50 value of 37 nM, and displays weaker inhibition toward PRMT6, with an IC50...		Histone Methyltransferase