Home Tools
Log in
Cart

Search Result

Search Results for " plk1/brd4-in-1 "

2

Compounds

Cat No. Product Name Synonyms Targets
T64058 PLK1/BRD4-IN-1
PLK1/BRD4-IN-1 (9b) is an orally active dual inhibitor of PLK1 (IC50: 22 nM) and BRD4 (IC50: 109 nM). It has been shown to have good anti-tumour effects in vivo.
T79065 WWL0245 Epigenetic Reader Domain
WWL0245 is a potent and selective BRD4-targeting PROTAC that exhibits sub-nanomolar degradation efficiency (DC50 < 1 nM) for BRD4 over BRD2/3 and PLK1 (DC50 > 1 μM). It demonstrates pronounced selective cytotoxicity in B...
TargetMol