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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
TP1957 | PKI(5-24) | PKI (5-24) | |
High affinity PKA inhibitor (Ki = 2.3 nM). | |||
TP1957L | PKI (5-24) Acetate(99534-03-9 free base) | PKA | |
PKI (5-24) Acetate is a high affinity PKA inhibitor (Ki = 2.3 nM). | |||
T76482 | PKI (5-24),amide | ||
PKI (5-24),amide (IP20-amide) is a potent inhibitor of cAMP-dependent protein kinase (PKA) (PKA), with an inhibition constant (K i ) of 2.3 nM [1]. This 20-residue peptide mirrors the active segment of the heat-stable in... | |||
T75739 | PKI(5-24) TFA | ||
PKI(5-24) TFA is a synthetic peptide inhibitor of PKA (cAMP-dependent protein kinase), characterized by its potent and competitive inhibition properties, exhibiting a K i of 2.3 nM. It corresponds to residues 5-24 found ... | |||
T4978 | Sarpogrelate hydrochloride | MCI-9042 | 5-HT Receptor |
Sarpogrelate hydrochloride (MCI-9042) , a selective 5-HT2 antagonist, has been widely used as an anti-platelet agent for the treatment of PAD. Target: 5-HT2 Recepter Sarpogrelate is a drug which acts as an antagonist at ... | |||
T36019 | PKA Inhibitor (5-24) (trifluoroacetate salt) | ||
PKI PKA Inhibitor (5-24) is a synthetic peptide inhibitor of PKA (cAMP-dependent protein kinase) (Ki= 2.3 nM) derived from the active site of the skeletal muscle inhibitor protein.1It mimics the protein substrate by bind... | |||
T36084 | PKI-179 | ||
PKI-179 is a potent, orally active compound that functions as a dual PI3K/mTOR inhibitor. It demonstrates IC50 values of 8 nM for PI3K-α, 24 nM for PI3K-β, 74 nM for PI3K-γ, 77 nM for PI3K-δ, and 0.42 nM for mTOR. Additi... |