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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T6905 | Netupitant | Ro 67-31898/000,CID 6451149 | Neurokinin receptor |
Netupitant (CID 6451149) is a specific neurokinin 1 (NK1) receptor antagonist (Ki: 0.95 nM). | |||
T12211 | Netupitant metabolite Monohydroxy Netupitant | Monohydroxy Netupitant | Others |
Monohydroxy Netupitant is a highly selective antagonist of NK1 receptor, and is Netupitant metabolite. | |||
T12212 | Netupitant metabolite N-desmethyl Netupitant | N-desmethyl Netupitant | Others |
N-desmethyl Netupitant is a highly selective antagonist of NK1 receptor, and is Netupitant metabolite. | |||
T12213 | Netupitant metabolite Netupitant N-oxide | Netupitant N-oxide | Others |
Netupitant N-oxide is a highly selective antagonist of NK1 receptor, is Netupitant metabolite. | |||
T19434 | Monohydroxy Netupitant D6 | Others | |
Monohydroxy Netupitant D6 is a metabolite of Netupitant. | |||
T12210 | Netupitant D6 | CID-6451149 D6 | Others |
Netupitant D6 is the deuterium labeled Netupitant, which is a selective and orally active antagonist of neurokinin-1 receptor. | |||
T19474 | Netupitant N-oxide D6 | Others | |
Netupitant N-oxide D6 is a Netupitant metabolite, is the deuterium labeled Netupitant N-oxide. | |||
T19452 | N-desmethyl Netupitant D6 | Others | |
N-desmethyl Netupitant D6 is the deuterium labeled N-desmethyl Netupitant, which is a Netupitant metabolite. | |||
T15341 | Fosnetupitant | Pronetupitant | Others |
Fosnetupitant is a methylene phosphate prodrug of Netupitant. It has a pKi of 9.5 for the human NK1 receptor. | |||
T78104 | Fosnetupitant chloride monohydrochloride | Pronetupitant chloride monohydrochloride | Neurokinin receptor |
Fosnetupitant chloride monohydrochloride (Pro-netupitant chloride monohydrochloride) is a selective NK1 antagonist exhibiting high affinity for the human NK1 receptor with a pK i value of 9.5, and a lower affinity for th... | |||
T9735 | 6-(4-methylpiperazin-1-yl)-4-o-tolylnicotinamide | Others | |
6-(4-methylpiperazin-1-yl)-4-o-tolylnicotinamide can be used in the synthesis of befetupitant and netupitant. |