Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Fosnetupitant is a methylene phosphate prodrug of Netupitant. It has a pKi of 9.5 for the human NK1 receptor.
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
25 mg | 6-8 weeks | $ 1,520.00 | |
50 mg | 6-8 weeks | $ 1,980.00 | |
100 mg | 6-8 weeks | $ 2,500.00 |
Description | Fosnetupitant is a methylene phosphate prodrug of Netupitant. It has a pKi of 9.5 for the human NK1 receptor. |
In vitro | Fosnetupitant shows a micromolar affinity for the 5-HT6 (pKi ~ 5.2) receptor and type L Ca2+ channels (pKi ~ 5.7). However, it does not bind all the other proteins investigated. |
In vivo | After i.v. injection in rats, Pronetupitant is rapidly and extensively converted to Netupitant. |
Synonyms | Pronetupitant |
Molecular Weight | 688.6 |
Formula | C31H35F6N4O5P |
CAS No. | 1703748-89-3 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
You can also refer to dose conversion for different animals. More
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Fosnetupitant 1703748-89-3 Others Pronetupitant inhibitor inhibit