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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T2325 | Neratinib | HKI-272 | EGFR , HER |
Neratinib (HKI-272) (HKI-272) is an orally available, irreversible tyrosine kinase inhibitor for HER2 and EGFR (IC50: 59/92 nM), respectively. | |||
T67385 | Neratinib maleate | HKI-272 maleate | EGFR , HER |
Neratinib maleate (HKI-272 maleate) is an irreversible, orally active and highly selective inhibitor of HER2 and EGFR with IC50 values of 59 nM and 92 nM, respectively.Neratinib maleate has antitumor activity and can be ... | |||
T71387 | Neratinib maleate monohydrate | ||
Neratinib maleate monohydrate is an irreversible inhibitor of the HER-2 receptor tyrosine kinase with potential antineoplastic activity. | |||
T70829 | Neratinib pyridine N-oxide | ||
Neratinib pyridine N-oxide is an irreversible inhibitor of the HER-2 receptor tyrosine kinase with potential antineoplastic activity. | |||
T70830 | Neratinib dimethylamine N-oxide | ||
Neratinib dimethylamine N-oxide is an irreversible inhibitor of the HER-2 receptor tyrosine kinase with potential antineoplastic activity. | |||
T70828 | HBY-793 | ||
HBY-793 is an HIV-1 proteinase inhibitor. | |||
T70827 | MDL-102234 | ||
MDL-102234 is an adenosine A1 receptor antagonist. |