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Search Results for " mk0457 "

2

Compounds

Cat No. Product Name Synonyms Targets
T2509 Tozasertib MK-0457,VX 680 Aurora Kinase , Autophagy
Tozasertib (MK-0457) is a pan-Aurora kinase inhibitor (Kis: 0.6/18/4.6 nM for Aurora A/Aurora B/Aurora C). It shows selectivity against more than 190 different kinases.
T68415 Tozasertib lactate
Tozasertib lactate is a potent and selective small-molecule inhibitor of the Aurora kinases which suppresses tumor growth by inducing apoptosis in tumor cells in which Aurora kinases are overexpressed.
TargetMol