20
Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
TP1895L1 | KYL acetate(676657-00-4 free base) | Ephrin Receptor | |
KYL acetate is an EphA4 receptor tyrosine kinase inhibitor (Kd = 0.8 μM); inhibits EphA4-EphrinA5 interactions (IC50 = 6.34 μM). Prevents AβO induced synaptic damage, dendritic spine loss and prevents the blocking of LTP... | |||
TP1895 | KYL peptide | KYL | |
KYL peptide is an EphA4 receptor tyrosine kinase inhibitor (Kd = 0.8 μM); inhibits EphA4-EphrinA5 interactions (IC50 = 6.34 μM). Prevents AβO induced synaptic damage, dendritic spine loss and prevents the blocking of LTP... | |||
T0604 | Desalkylterbuthylazine | Others | |
Desalkylterbuthylazine is used as pharmaceutical intermediates. | |||
T40030 | Thalidomide 4'-ether-alkylC2-amine hydrochloride | halidomide-linker 6 | E3 Ligase Ligand-Linker Conjugate |
Thalidomide 4'-ether-alkylC2-amine hydrochloride (halidomide-linker 6) is a synthesized E3 ligase ligand-linker conjugate. | |||
T36282 | VH 032 amide-alkylC7-amine | VH 032 amide-alkylC7-amine | |
Functionalized von-Hippel-Lindau protein ligand (VHL) for PROTAC research and development; incorporates an E3 ligase ligand plus an alkyl linker ready for conjugation to a target protein ligand. Part of a range of funct... | |||
T36276 | Thalidomide 4'-oxyacetamide-alkylC8-amine | Thalidomide 4'-oxyacetamide-alkylC8-amine | |
Functionalized cereblon ligand for PROTAC research and development; incorporates an E3 ligase ligand plus an alkylC8 linker with terminal amine ready for conjugation to a target protein ligand. Part of a range of functi... | |||
T36250 | Thalidomide 4'-oxyacetamide-alkylC1-PEG3-alkylC3-amine | Thalidomide 4'-oxyacetamide-alkylC1-PEG3-alkylC3-amine | |
Functionalized cereblon ligand for PROTAC research and development; incorporates an E3 ligase ligand plus an alkylC1-PEG3-alkylC3 linker with terminal amine ready for conjugation to a target protein ligand. Part of a ra... | |||
T36270 | (S,R,S)-AHPC-phenol-alkylC6-amine dihydrochloride | VH 032 phenol-alkylC6-amine | |
Functionalized von-Hippel-Lindau (VHL) protein ligand for PROTAC research and development; incorporates an E3 ligase ligand plus an alkyl linker ready for conjugation to a target protein ligand. Part of a range of funct... | |||
T70854 | Protokylol hydrochloride | ||
Protokylol hydrochloride is the salt form of Protokylol (free base) (Asmetil, Caytine, Palison, Ventaire), a β-adrenergic receptor agonist used as a bronchodilator in Europe and the United States. It is methylenedioxyphe... | |||
T39876 | Thalidomide 4'-oxyacetamide-alkyl-C2-amine hydrochloride | Thalidomide 4'-oxyacetamide-alkyl-C2-amine hydrochloride | |
Thalidomide 4'-oxyacetamide-alkyl-C2-amine hydrochloride consists of a cereblon (CRBN) ligand for the E3 ubiquitin ligase and a linker, making it suitable for PROTACs design. | |||
T83954 | VH 032 amide-alkylC7-acid | (S,R,S)-AHPC-amido-C7-acid | |
VH 032 amide-alkylC7-acid is a specialized compound designed for PROTAC research and development, serving as a functionalized von-Hippel-Lindau (VHL) protein ligand. It combines an E3 ligase ligand with an alkylC7 linker... | |||
T18306 | MC-Alkyl-Hydrazine Modified MMAF | Others | |
MC-Alkyl-Hydrazine Modified MMAF is a potent antitumor drug-linker conjugate for ADC, incorporating Modified MMAF, a tubulin inhibitor, through a noncleavable MC-Alkyl-Hydrazine linkage[1]. | |||
T74372 | N-Desalkyludenafil | ||
N-Desalkyludenafil, a metabolite of Udenafil, functions as a PDE5 inhibitor and is utilized in the study of erectile dysfunction [1]. | |||
T36279 | VH 032 amide-alkylC3-amine | VH 032 amide-alkylC3-amine | |
Functionalized von-Hippel-Lindau (VHL) protein ligand for PROTAC research and development; incorporates an E3 ligase ligand plus an alkyl C3 linker and terminal amine ready for conjugation to a target protein ligand. Pa... | |||
T36274 | VH 101 phenol-alkylC6-amine | VH 101 phenol-alkylC6-amine | |
Functionalized von-Hippel-Lindau protein ligand (VHL) for PROTAC research and development; incorporates an E3 ligase ligand plus an alkylC6 linker with terminal amine ready for conjugation to a target protein ligand. Pa... | |||
T36263 | Pomalidomide 4'-alkylC8-acid | Pomalidomide 4'-alkylC8-acid | |
Functionalized cereblon ligand for PROTAC research and development; incorporates an E3 ligase ligand plus an alkylC8 linker with terminal acid ready for conjugation to a target protein ligand. Part of a range of functio... | |||
T36273 | VH 101 phenol-alkylC4-amine | VH 101 phenol-alkylC4-amine | |
Functionalized von-Hippel-Lindau protein ligand (VHL) for PROTAC research and development; incorporates an E3 ligase ligand plus an alkylC4 linker with terminal amine ready for conjugation to a target protein ligand. Pa... | |||
T40053 | Boc-A 410099.1 amide-alkylC4-amine | Boc-A 410099.1 amide-alkylC4-amine | |
Boc-A 410099.1 amide-alkylC4-amine is a functionalized IAP ligand for PROTACs, comprising of an IAP ligand and an amide-alkylC4 linker terminating in an amine group. It has the ability to form conjugates with target prot... | |||
T83961 | Thalidomide 5'-amine-alkylC6-amine | ||
Thalidomide 5'-amine-alkylC6-amine serves as a specialized cereblon ligand for PROTAC research and development, combining an E3 ligase ligand and an alkylC6 linker with a terminal amine for target protein ligand conjugat... | |||
T34865 | Thyminalkylamine | ||
Thyminalkylamine is a biochemical. |