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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T21069 | Lumateperone | ITI 722,ITI722,ITI-007,ITI007 | 5-HT Receptor |
Lumateperone (ITI 722) is a 5HT2A receptor antagonist and a dopamine receptor phosphoprotein modulator (DPPM). | |||
TQ0084 | Lumateperone Tosylate | ITI-007 | Dopamine Receptor , 5-HT Receptor |
lumateperone Tosylate (ITI-007) is a 5-HT2A receptor antagonist (Ki: 0.54 nM), a SERT blocker (Ki: 61 nM), a partial agonist of presynaptic D2 receptors and an antagonist of postsynaptic D2 receptors (Ki: 32 nM). |