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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T22748 | DQP 1105 | NMDAR | |
DQP 1105 is a NMDA receptor antagonist. | |||
T16801 | (RS)-(Tetrazol-5-yl)glycine | LY 285265,D,L-(tetrazol-5-yl)glycine | NMDAR , iGluR |
(RS)-(Tetrazol-5-yl)glycine (LY 285265) (D,L-(tetrazol-5-yl)glycine) is an effective and selective N-methyl-D-aspartate receptor agonist. (RS)-(Tetrazol-5-yl)glycine has EC50s of 99 nM, 1.7 μM for GluN1/GluN2D, and GluN1... | |||
T15407 | GNE-0723 | Others | |
GNE 0723 is an NMDAR brain permeable positive allosteric modulator (EC50: 21 nM for GluN2A; 7.4 and 6.2 μM for GluN2C and GluN2D, respectively). | |||
T15408 | GNE 5729 | Others | |
GNE 5729 is an NMDAR of brain permeable positive allosteric modulator (EC50: 37 nM for GluN2A; 4.7 and 9.5 μM for GluN2C and GluN2D, respectively). | |||
T61227 | NAB-14 | ||
NAB-14 is a powerful and selective chemical compound that acts as a non-competitive antagonist for GluN2C and GluN2D receptors. With an IC50 value of 580 nM for GluN1/GluN2D, NAB-14 demonstrates high potency. This compou... | |||
T24551 | NSC339614 potassium | NSC 339614 potassium,NSC-339614 potassium,NSC339614 potassium salt | |
NSC339614 potassium is a selective GluN1/GluN2C and GluN1/GluN2D receptors potentiator. | |||
T19881 | UBP608 | UBP-608,UBP 608 | |
UBP608 is an allosteric modulator of NMDA receptor family. It selectively inhibits GluN1/GluN2A receptors with a 23-fold selectivity compared to GluN1/GluN2D receptors. | |||
T73491 | TP-050 | ||
TP-050 is a potent, selective NMDAR agonist that is orally active, showing EC50 values of 0.51 µM for GluN2A and 9.6 µM for GluN2D. This compound can cross the blood-brain barrier (BBB), enhancing hippocampal long-term (... | |||
T79611 | DQP-26 | iGluR | |
DQP-26, a potent negative allosteric modulator of NMDA receptors (NMDARs), exhibits IC50 values of 0.77 μM for GluN2C and 0.44 μM for GluN2D subunits, indicating potential application in research on NMDAR-associated neur... |