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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T11384 | Gefitinib-d8 | ZD1839 D8,Gefitinib D8 | Others |
Gefitinib is an EGFR tyrosine kinase inhibitor, with IC50 of 2-37 nM in NR6wtEGFR cells. Gefitinib D8 is a deuterium labeled Gefitinib. | |||
T19489 | O-Desmethyl gefitinib D8 | EGFR | |
O-Desmethyl gefitinib D8 is a deuterium labeled O-Desmethyl gefitinib that is an active metabolite of Gefitinib in human plasma. | |||
TMIH-0402 | O-Desmethyl Gefitinib-d8 | ||
O-Desmethyl Gefitinib-d8 is a deuterated compound of O-Desmethyl Gefitinib. O-Desmethyl Gefitinib has a CAS number of 847949-49-9. O-Desmethyl gefitinib inhibits EGFR (IC50: 36 nM in subcellular assays). In human plasma,... |