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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T6021 | GSK1324726A | I-BET726 | Apoptosis , Epigenetic Reader Domain |
GSK1324726A (I-BET726) is a greatly specific inhibitor of BET family proteins for BRD2(IC50=41 nM), BRD3(IC50=31 nM), and BRD4 (IC50=22 nM). |