2
Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T31936 | GLL398 | GLL 398,GLL-398 | |
GLL398 is an oral selective estrogen receptor down-regulating agent that strongly binds to ERα (IC50 =1.14 nM) and effectively degrades ERα in MCF-7 breast cancer cells (IC50 = 0.21 μM). | |||
T9997 | GLL 398 | Estrogen Receptor/ERR | |
GLL 398 is an orally active and selective degrader of estrogen receptor with an IC50 of 1.14 nM. GLL 398 blocks tumor growth in xenograft breast cancer models. |