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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T11393 | GET73 | Gamma hydroxybutyric acid analogue,GET 73 | GluR |
GET73 (Gamma hydroxybutyric acid analogue) is an negative allosteric modulator of mGluR5. GET73 is a naturally occurring neurotransmitter. GET73 has anti-alcohol and anxiolytic properties. | |||
T5273 | 2-Hydroxy-3-methylbutanoic acid | 2-Hydroxy-3-methylbutyric acid,2-Hydroxyisovaleric Acid,(±)-2-Hydroxyisopentanoic Acid | Others , Endogenous Metabolite |
2-Hydroxy-3-methylbutanoic acid ((±)-2-Hydroxyisopentanoic Acid) is a metabolite found in the urine of patients with phenylketonuria, methylmalonic acidemia, propionic acidemia, 3-ketothiolase deficiency, isovaleric acid... | |||
T23473 | Trans-4-Hydroxycrotonic acid | Others | |
ligand of γ-hydroxybutyric acid (GHB) receptor | |||
T69259 | NCS-356 sodium | ||
NCS-356 sodium is a GHB receptor agonist. | |||
T39962 | Valiloxibic acid | XWL-008,Acidum valiloxibicum | |
Valiloxibic acid is a prodrug of γ-Hydroxybutyric acid (GHB).GHB is a naturally occurring neurotransmitter and a psychoactive drug, it acts on the GHB receptor and is a weak agonist at the GABAB receptor. | |||
T24146 | HOCPCA | ||
HOCPCA is an effective and selective ligand for the GHB binding sites that acts by binding with 27 times better affinity than GHB itself and crossing the blood-brain barrier in vitro and in vivo. | |||
T68181 | NCS-356 | ||
NCS-356 is a GHB receptor agonist. | |||
T71533 | NCS-356 sodium monohydrate | ||
NCS-356 sodium monohydrate is a GHB receptor agonist. | |||
T29058 | UMB68 sodium | UMB-68 sodium,UMB68,UMB-68,UMB 68 | |
UMB-68 is a GHB receptor ligand with no affinity (IC(50) >100 microM) at GABA(A) or GABA(B) receptors. | |||
T37822 | AR-C 141990 hydrochloride | ||
Monocarboxylate transporter (MCT1) inhibitor (pKi = 7.6. Exhibits approximately 10-fold selectivity for MCT1 over MCT2 and no significant activity against MCT3 or 4. Inhibits graft versus host response and prolongs card... |