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Search Results for " difelikefalin "

6

Compounds

Cat No. Product Name Synonyms Targets
T38419 Difelikefalin CR-845,FE-202845
Difelikefalin (CR-845; FE-202845) is a peripherally restricted, selective agonist of the kappa opioid receptor (KOR). It exhibits anti-inflammatory properties and holds promise for modulating pruritus in conditions assoc...
TP2501 Difelikefalin acetate Difelikefalin acetate(1024828-77-0 free base),CR 845 acetate,FE 202845 acetate Opioid Receptor
Difelikefalin acetate (CR 845 acetate) is a peripherally restricted kappa opioid receptor agonist. CR845 exhibit low P450 CYP inhibition and low penetration into the brain.
TP2485 difelikefalin acetate(1024828-77-0 Free base) Opioid Receptor
is a ketone and a building block.
T69537 Difelikefalin HCl
Difelikefalin HCl is a κ-opioid receptor (KOR) agonist. It activates KOR in HEK293 cells expressing the human receptor (EC50 = 0.16 nM in a transactivation assay) and inhibits forskolin-induced cAMP production in R1.G1 m...
T37483 Difelikefalin (trifluoroacetate salt)
Difelikefalin is a κ-opioid receptor (KOR) agonist.1It activates KOR in HEK293 cells expressing the human receptor (EC50= 0.16 nM in a transactivation assay) and inhibits forskolin-induced cAMP production in R1.G1 mouse ...
T69530 Difelikefalin TFA
Difelikefalin TFA is a κ-opioid receptor (KOR) agonist. It activates KOR in HEK293 cells expressing the human receptor (EC50 = 0.16 nM in a transactivation assay) and inhibits forskolin-induced cAMP production in R1.G1 m...
TargetMol