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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T36061 | N-Desmethyl Sildenafil | Desmethylsildenafil,UK-103,320 | Drug Metabolite |
N-Desmethyl Sildenafil (UK-103,320) (Desmethylsildenafil) is a prominent metabolite of Sildenafil, a potent inhibitor of phosphodiesterase type 5 (PDE5). | |||
T36062 | N-Desmethyl Sildenafil (citrate) | ||
N-Desmethyl sildenafil is a major metabolite of sildenafil . N-Desmethyl sildenafil is formed via oxidative metabolism of sildenafil by the cytochrome (CYP) P450 isoforms CYP3A4, CYP3A5, and CYP3A7. |