2
Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T14990 | CDK12-IN-3 | CDK | |
CDK12-IN-3 is a selective CDK12 inhibitor (IC50: 491 nM in an enzymatic assay). | |||
T62926 | CDK7/12-IN-1 | ||
CDK7/12-IN-1 is a selective inhibitor of CDK7/12, acting on CDK7 (IC50: 3 nM) and CDK 12 (IC50: 277 nM). Inhibition of CDK7 and CDK12 is an effective inhibitor of tumour growth. |