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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T10623 | BSH-IN-1 | Potassium Channel | |
BSH-IN-1 is a potent and covalent inhibitor of gut bacterial recombinant bile salt hydrolases (BSHs; IC50s: 108 nM and 427 nM for B. longum BSH and B. theta BSH). | |||
T11515 | Gut restricted-7 | GR-7 | Potassium Channel |
Gut restricted-7 (GR-7) (GR-7) is a covalent and orally active pan-bile salt hydrolase (BSH) inhibitor. It decreases gut bacterial BSHs and decreases deconjugated bile acid levels in the feces of mice. | |||
T63616 | AAA-10 formic | ||
AAA-10 formic is an orally active inhibitor of intestinal bacterial bile salt hydrolase (BSH) against B. thetarBSH (IC50: 10 nM) and B. longumrBSH (IC50: 80 nM). | |||
T63060 | AAA-10 | ||
AAA-10 is an orally active inhibitor of bile salt hydrolase (BSH) in B. intestinalis that acts on B. thetarBSH (IC50: 10 nM) and B. longumrBSH (IC50: 80 nM). |