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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T10350 | Apremilast-d5 | Apremilast D5,CC-10004 D5 | TNF , PDE |
Apremilast D5 (CC-10004 D5) is a deuterium-labeled Apremilast. Apremilast is an orally available inhibitor of PDE-4 (IC50: 74 nM). Apremilast inhibits TNF-α release by lipopolysaccharide (IC50: 104 nM). | |||
T12656 | (Rac)-Apremilast D5 | (Rac)-CC-10004 D5 | Others |
(Rac)-Apremilast D5 is a deuterium-labeled version of the enantiomer (R)-Apremilast, also known as (R)-CC-10004, which itself is one specific form of Apremilast. |