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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T7656 | Apelin-13 | ||
Apelin-13 is a 13-amino acid peptide sequence found in the central and peripheral nervous system that is an endogenous ligand for the G protein-coupled receptor angiotensin II protein J (APJ), with an EC50 value of 0.37 ... | |||
TP1260 | [Pyr1]-Apelin-13 | [pGlu1]-Apelin-13 | Apelin receptor |
[Pyr1]-Apelin-13 ([pGlu1]-Apelin-13) is a potent and selective endogenous Apelin receptor (APJ) agonist. | |||
T7847 | Apelin-13 triTFA(217082-58-1(free base)) | Others | |
Apelin-13 triTFA is the endogenous ligand of the APJ receptor, activating this G protein-coupled receptor with an EC50 value of 0.37 nM. | |||
T35374 | (Ala13)-Apelin-13 | (Ala13)-Apelin-13 | Others |
(Ala13)-Apelin-13 is a useful organic compound for research related to life sciences. The catalog number is T35374 and the CAS number is 568565-11-7. | |||
T35374L | (Ala13)-Apelin-13 acetate | Apelin receptor | |
(Ala13)-Apelin-13 acetate, an APJ antagonist, modulates CRF-induced enhanced colonic motility, visceral sensation, and gut barrier. | |||
TP1424 | Apelin-13 TFA (217082-58-1 free base) | Apelin-13 TFA | |
Apelin-13 is an endogenous ligand of APJ receptor, and the EC 50 value of activated G protein coupled receptor is 0.37 nM. | |||
T78109 | (Ala13)-Apelin-13 TFA | ||
'(Ala13)-Apelin-13 TFA acts as a potent antagonist of the apelin receptors (APJ) and impedes gastric motility via the vagal cholinergic pathway [1].' | |||
T4390 | ML221 | Apelin receptor , Arrestin | |
ML221 is a potent apelin /APJ functional antagonist, inhibiting apelin-13-mediated activation of APJ, with IC50s of 0.70 μM in the cAMP assay, and 1.75 μM in the β-arrestin assay, and EC80 of 10 nM in both assays. | |||
TP2001 | MM 54 | ||
Potent apelin receptor antagonist (Ki = 82 nM; IC50 = 93 nM). Antagonizes the inhibitory affect of [Pyr1]-Apelin-13 on forskolin-induced cAMP accumulation in CHO-K1-APJ cells. Recuces tumor expansion and lengthens surviv... | |||
T39813 | APJ receptor agonist 1 | ||
APJ receptor agonist 1, a potent biphenyl acid derivative, acts as an agonist (EC50 of 0.093 nM and 0.12 nM for human and rat APJ receptors, respectively) for the APJ receptor (APJ-R). It exhibits significant in vitro po... |