4
Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T7609 | ARS-1620 | Ras | |
ARS-1620 is a covalent inhibitor of K-RASG12C. | |||
T22249 | 1588-A4 | ARS-1620 Intermediate | Ras |
1588-A4 (ARS-1620 Intermediate) is an intermediate of ARS-1620 which is an atropisomeric selective KRASG12C inhibitor with desirable pharmacokinetics. | |||
T10375 | ARS-1323 | Ras | |
ARS-1323 is the racemate of ARS-1620 and a mutant K-ras G12C inhibitor. | |||
T10376 | ARS-1630 | Ras | |
ARS-1630 is a mutant K-ras G12C inhibitor. It is a less active enantiomer of ARS-1620. |