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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T68415 | Tozasertib lactate | ||
Tozasertib lactate is a potent and selective small-molecule inhibitor of the Aurora kinases which suppresses tumor growth by inducing apoptosis in tumor cells in which Aurora kinases are overexpressed. | |||
T2509 | Tozasertib | MK-0457,VX 680 | Aurora Kinase , Autophagy |
Tozasertib (MK-0457) is a pan-Aurora kinase inhibitor (Kis: 0.6/18/4.6 nM for Aurora A/Aurora B/Aurora C). It shows selectivity against more than 190 different kinases. |