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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T5398 | BMS 599626 2HCl (873837-23-1(HCl)) | AC480 dihydrochloride | HER |
BMS 599626 2HCl (873837-23-1(HCl)) (AC480 dihydrochloride) is a selective inhibitor of HER1 and HER2 (IC50s: 20 nM and 30 nM), ~8-fold less potent to HER4, >100-fold to Lck, VEGFR2, c-Kit, MET, etc. | |||
T5390 | BMS-599626 Hydrochloride | AC480 Hydrochloride | HER |
BMS-599626 Hydrochloride (AC480 Hydrochloride) is an orally bioavailable inhibitor of the HER1, HER2 and HER4 tyrosine kinases (IC50 =22, 32 and 190 nM, respectively) with potential antineoplastic activity. BMS-599626 Hy... |