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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T2344 | LY 344864 | LY344864 | 5-HT Receptor |
LY 344864, a specifc receptor agonist, is an affinity of 6 nM (Ki) at the recently cloned 5-HT1F receptor. | |||
T2344L | LY 344864 racemate | 5-HT Receptor | |
LY 344864 racemate is a 5-HT1F receptor agonist. | |||
T4266 | LY334370 | LY 334370 | 5-HT Receptor |
LY334370 is a selective 5-HT1F receptor agonist with a Ki of 1.6 nM | |||
T4118 | SB 271046 hydrochloride | SB 271046A | 5-HT Receptor |
SB 271046 hydrochloride (SB 271046A) is selective, orally active 5-HT6 antagonist (pKi values are 9.02-8.92, 6.35, 6.55, 6.27 at 5-HT6, 5-HT1A, 5-HT1D and D3, and 6.05, 5.95, 5.76, 5.73, 5.62, 5.55, 5.41, 5.39, 5.27 and ... | |||
T1092 | Zolmitriptan | 311C90,BW-311C90 | 5-HT Receptor |
Zolmitriptan (311C90) selectively binds to and activates serotonin (5-HT) 1B receptors expressed in intracranial arteries and 5-HT 1D receptors located on peripheral trigeminal sensory nerve terminals in the meninges and... | |||
T27059 | CP-122288 | ||
CP-122288 is a potent and selective agonist for the 5-HT1B, 5-HT1D and 5-HT1F serotonin receptor subtypes. CP-122288 is potent as an inhibitor of plasma protein extravasation and neurogenic inflammation. | |||
T22952 | LY 334370 hydrochloride | Others | |
5-HT1F receptor agonist | |||
T11902 | LY 344864 S-enantiomer | Others | |
LY 344864 S-enantiomer, the S-enantiomer of LY344864, serves as a 5-HT1F receptor agonist. | |||
T27915 | LY 302148 | LY-302148,LY302148 | |
LY 302148 , a 5-HT1F receptor agonist, inhibits neurogenic dural inflammation in guinea pigs. It has potential for migraine therapeutics. | |||
T41295 | LY 344864 hydrochloride | ||
LY 344864 hydrochloride is a selective receptor agonist with an affinity of 6 nM (Ki) at the 5-HT1F receptor. | |||
T2459 | BRL 54443 | BRL54443 | 5-HT Receptor |
BRL 54443 is a potent 5-HT1E/1F receptor agonist (pKi values are 8.7 and 8.9 respectively). | |||
T19690 | SB 224289 | SB224289,SB-224289 | |
SB 224289 is a selective antagonist of 5-HT1B receptor with pKi of 8.2. It is a centrally active following oral administration in vivo. SB 224289 displays 60-fold selectivity over 5-HT1D, 5-HT1A, 5-HT1E, 5-HT1F, 5-HT2A a... |