Powder: -20°C for 3 years | In solvent: -80°C for 1 year
SB 224289 is a selective antagonist of 5-HT1B receptor with pKi of 8.2. It is a centrally active following oral administration in vivo. SB 224289 displays 60-fold selectivity over 5-HT1D, 5-HT1A, 5-HT1E, 5-HT1F, 5-HT2A and 5-HT2C receptors in radioligand binding and functional assays.
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
25 mg | 10-14 weeks | $ 2,270.00 | |
50 mg | 10-14 weeks | $ 2,980.00 | |
100 mg | 10-14 weeks | $ 4,000.00 |
Description | SB 224289 is a selective antagonist of 5-HT1B receptor with pKi of 8.2. It is a centrally active following oral administration in vivo. SB 224289 displays 60-fold selectivity over 5-HT1D, 5-HT1A, 5-HT1E, 5-HT1F, 5-HT2A and 5-HT2C receptors in radioligand binding and functional assays. |
Synonyms | SB224289, SB-224289 |
Molecular Weight | 520.62 |
Formula | C32H32N4O3 |
CAS No. | 180083-23-2 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: Soluble
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SB 224289 180083-23-2 SB224289 SB-224289 inhibitor inhibit