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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T81375 | PROTAC TTK degrader-1 | PROTACs | |
PROTAC TTK degrader-1, a potent threonine tyrosine kinase (TTK) PROTAC degrader, demonstrates DC50 values of 1.7 nM in COLO-205 cells and 5.8 nM in HCT-116 cells, indicating effective target degradation. Furthermore, it ... |