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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T79167 | BET-IN-15 | Epigenetic Reader Domain | |
BET-IN-15 (compound 1) is a potent, orally active inhibitor of BET, demonstrating inhibitory IC50 values of 0.64 nM for BRD4-BD1 and 0.25 nM for BRD4-BD2. It exhibits antiproliferative activity [1]. |