Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Zaldaride maleate inhibits CaM (calmodulin)-stimulated cAMP phosphodiesterase activity (IC50: 3.3 nM). Zaldaride maleate is an effective and selective inhibitor of calmodulin. Zaldaride maleate prevents estrogen-induced transcription activation by ER, reversibly blocks voltage-activated Na+, Ca2+, and K+ currents in PC12 cells and inhibits nAChR.
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
1 mg | 35 days | $ 93.00 | |
5 mg | 35 days | $ 290.00 | |
10 mg | 35 days | $ 488.00 | |
25 mg | 35 days | $ 993.00 |
Description | Zaldaride maleate inhibits CaM (calmodulin)-stimulated cAMP phosphodiesterase activity (IC50: 3.3 nM). Zaldaride maleate is an effective and selective inhibitor of calmodulin. Zaldaride maleate prevents estrogen-induced transcription activation by ER, reversibly blocks voltage-activated Na+, Ca2+, and K+ currents in PC12 cells and inhibits nAChR. |
Targets&IC50 | Calmodulin:3.3 nM |
Synonyms | CGS-9343B, KW 5617 |
Molecular Weight | 544.6 |
Formula | C30H32N4O6 |
CAS No. | 109826-27-9 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
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Zaldaride maleate 109826-27-9 Others KW5617 KW-5617 CGS-9343B KW 5617 Zaldaride Maleate inhibitor inhibit