Powder: -20°C for 3 years | In solvent: -80°C for 1 year
ZEN-3219 is a BET inhibitor, which has inhibitory effect on BRD4(BD1), BRD4(BD2) and BRD4(BD1BD2). ZEN-3219 has inhibitory effect on BRD4(BD1), The IC50 values of BRD4(BD2) and BRD4(BD1BD2) were 0.48, 0.16 and 0.47 μM, respectively. ZEN-3219 is a component of PROTAC molecule and can induce BRD4 degradation.
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
1 mg | In stock | $ 132.00 | |
5 mg | In stock | $ 328.00 | |
10 mg | In stock | $ 528.00 | |
25 mg | In stock | $ 955.00 | |
50 mg | In stock | $ 1,390.00 | |
100 mg | In stock | $ 1,880.00 | |
500 mg | In stock | $ 3,780.00 |
Description | ZEN-3219 is a BET inhibitor, which has inhibitory effect on BRD4(BD1), BRD4(BD2) and BRD4(BD1BD2). ZEN-3219 has inhibitory effect on BRD4(BD1), The IC50 values of BRD4(BD2) and BRD4(BD1BD2) were 0.48, 0.16 and 0.47 μM, respectively. ZEN-3219 is a component of PROTAC molecule and can induce BRD4 degradation. |
Targets&IC50 | BRD4 BD2:0.16 μM, BRD4 BD1/2:0.47 μM, BRD4 BD1:0.48 μM |
Molecular Weight | 322.36 |
Formula | C19H18N2O3 |
CAS No. | 1952264-34-4 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
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ZEN-3219 1952264-34-4 Chromatin/Epigenetic Others Epigenetic Reader Domain ZEN3219 ZEN 3219 inhibitor inhibit