Powder: -20°C for 3 years | In solvent: -80°C for 1 year
VU6015929 is an inhibitor of active dual discoidin domain receptor 1/2 (DDR1/2)( IC50s of 4.67 nM and 7.39 nM, respectively).
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
1 mg | In stock | $ 135.00 | |
5 mg | In stock | $ 289.00 | |
10 mg | In stock | $ 455.00 | |
25 mg | In stock | $ 753.00 | |
50 mg | In stock | $ 1,060.00 | |
100 mg | In stock | $ 1,430.00 | |
500 mg | In stock | $ 2,860.00 | |
1 mL * 10 mM (in DMSO) | In stock | $ 297.00 |
Description | VU6015929 is an inhibitor of active dual discoidin domain receptor 1/2 (DDR1/2)( IC50s of 4.67 nM and 7.39 nM, respectively). |
Targets&IC50 | DDR2:7.39 nM , DDR1:4.67 nM |
In vitro | VU6015929 potently blocks collagen-induced DDR1 activation and collagen-IV production, suggesting DDR1 inhibition as an exciting target for antifibrotic therapy[1]. |
Molecular Weight | 485.43 |
Formula | C24H19F4N5O2 |
CAS No. | 2442597-56-8 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 250 mg/mL (515.01 mM)
You can also refer to dose conversion for different animals. More
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VU6015929 2442597-56-8 Tyrosine Kinase/Adaptors Discoidin Domain Receptor (DDR) VU-6015929 VU 6015929 inhibitor inhibit