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USP7-IN-3

Catalog No. T13269 CAS 2202738-42-7

USP7-IN-3 is a potent and selective allosteric inhibitor of ubiquitin-specific <a href="/target/Protease" style="display: inline; color: #c13a36">Protease</a> 7 (USP7).

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USP7-IN-3, CAS 2202738-42-7

Pack Size	Availability	Price/USD
5 mg	10-12 weeks	$ 1,370.00
50 mg	10-12 weeks	$ 2,780.00
100 mg	10-12 weeks	$ 3,700.00

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Purity: 98%

Biological Description

Chemical Properties

Storage & Solubility Information

Description

USP7-IN-3 is a potent and selective allosteric inhibitor of ubiquitin-specific protease 7 (USP7).

Molecular Weight	568.59
Formula	C29H31F3N6O3
CAS No.	2202738-42-7

Storage

Powder: -20°C for 3 years

In solvent: -80°C for 2 years

Solubility Information

( < 1 mg/ml refers to the product slightly soluble or insoluble )

References and Literature

1. Gavory G, et al. Discovery and characterization of highly potent and selective allosteric USP7 inhibitors. Nat Chem Biol. 2018 Feb;14(2):118-125.

Related Products

Related compounds with same targets

USP8-IN-2 USP8-IN-3 USP15-IN-1 IMP-1710 HBX 41108 LDN-91946 FT827 USP7-IN-6

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Method for preparing in vivo formulation：Take μL DMSO master liquid, next add μL PEG300， mix and clarify, next add μL Tween 80，mix and clarify, next add μL ddH₂O, mix and clarify.

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Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.

Keywords

USP7-IN-3 2202738-42-7 Cell Cycle/Checkpoint DNA Damage/DNA Repair Ubiquitination DUB USP-7-IN-3 USP7IN3 USP7 IN 3 Inhibitor inhibitor inhibit

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