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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T13247 | UK-101 | UK101 , UK 101 | Proteasome |
UK-101 is a potent and selective inhibitor of the immunoproteasome LMP2, inhibiting β1i (LMP2), β1c (LMP2), and β5 (LMP2), with IC50s of 104 nM, 15 μM, and 1 μM. UK-101 has a 144-fold and 10-fold higher affinity for β1i ... |