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R 56865

Catalog No. T26016 CAS 104606-13-5

Synonyms: R-56865, R56865

R 56865 is a weak potential-operated channel inhibitor that inhibits the late sodium current in human isolated cardiomyocytes.

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R 56865, CAS 104606-13-5

Pack Size	Availability	Price/USD
1 mg	In stock	$ 293.00
5 mg	In stock	$ 722.00
10 mg	In stock	$ 987.00
25 mg	In stock	$ 1,520.00
50 mg	In stock	$ 1,980.00
100 mg	In stock	$ 2,500.00

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Purity: 99.08%

Biological Description

Chemical Properties

Storage & Solubility Information

Description

R 56865 is a weak potential-operated channel inhibitor that inhibits the late sodium current in human isolated cardiomyocytes.

Synonyms	R-56865, R56865
Molecular Weight	413.55
Formula	C23H28FN3OS
CAS No.	104606-13-5

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year

References and Literature

1. Wilhelm D,et al. Characterization of the interaction of R 56865 with cardiac Na- and L-type Ca channels. Br J Pharmacol. 1991 Oct;104(2):483-9. 2. Pijl AJ, et al. The negative inotropic and chronotropic effects of intravenous R 56865 during percutaneous transluminal coronary angioplasty. Br J Clin Pharmacol. 1995 May;39(5):531-5. 3. Verscheure Y,et al. Attenuation by R 56865, a novel cytoprotective drug, of regional myocardial ischemia- and reperfusion-induced electrocardiographic disturbances in anesthetized rabbits. J Cardiovasc Pharmacol. 1995 Jan;25(1):126-33. 4. Heers C,et al. Differential effect of R 56865 on ouabain binding to isolated sarcolemma and intact atrial tissue of guinea-pig. Br J Pharmacol. 1991 Mar;102(3):675-8.

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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.

Keywords

R 56865 104606-13-5 Membrane transporter/Ion channel Sodium Channel R-56865 R56865 inhibitor inhibit

Products are chemical reagents for research use only and are not intended for human use. We do not sell to patients.