Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Nerisopam is an agonist of gamma-aminobutyric acid (GABA) receptor.
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
1 mg | In stock | $ 142.00 | |
5 mg | In stock | $ 350.00 | |
10 mg | In stock | $ 530.00 | |
25 mg | In stock | $ 859.00 | |
50 mg | In stock | $ 1,180.00 | |
100 mg | In stock | $ 1,590.00 | |
500 mg | In stock | $ 3,190.00 | |
1 mL * 10 mM (in DMSO) | In stock | $ 475.00 |
Description | Nerisopam is an agonist of gamma-aminobutyric acid (GABA) receptor. |
In vivo |
Nerisopam application (30 mg/kg; 5 h; gastric cannula) cells in the reticular zone of the substantia nigra showed Fos-like immunopositivity.[6] Nerisopam (20 mg/kg;13 days; daily) for two weeks after a daily application, relatively weak Fos-like immunoreactivity was observed in the striatum and the subthalamic nucleus but not in the globus pallidus. Our results suggest that the striatal neurons are the primary targets of this anxiolytic and antipsychotic drug in the central nervous system.[6] |
Synonyms | EGIS-6775, GYKI 52322, GYKI52322, EGIS6775, GYKI-52322 |
Molecular Weight | 309.36 |
Formula | C18H19N3O2 |
CAS No. | 102771-12-0 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 25 mg/mL (41.38 mM)
You can also refer to dose conversion for different animals. More
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Nerisopam 102771-12-0 Membrane transporter/Ion channel Neuroscience GABA Receptor EGIS 6775 EGIS-6775 GYKI 52322 GYKI52322 EGIS6775 GYKI-52322 inhibitor inhibit