Powder: -20°C for 3 years | In solvent: -80°C for 1 year
LP-922761 is a potent, selective, and orally active AAK1 inhibitor with inhibitory effects on BMP-2 induced protein kinase (BIKE).
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
2 mg | In stock | $ 76.00 | |
5 mg | In stock | $ 129.00 | |
10 mg | In stock | $ 213.00 | |
25 mg | In stock | $ 382.00 | |
50 mg | In stock | $ 568.00 | |
100 mg | In stock | $ 813.00 | |
1 mL * 10 mM (in DMSO) | In stock | $ 143.00 |
Description | LP-922761 is a potent, selective, and orally active AAK1 inhibitor with inhibitory effects on BMP-2 induced protein kinase (BIKE). |
Targets&IC50 | AAK1:7.6 nM (cell assays), BIKE:24 nM, AAK1:4.8 nM (enzyme assays) |
In vivo | In mice, the brain-to-plasma ratio of LP-922761 was 0.007, indicating that LP-922761 was basically confined to the peripheral compartment[1]. |
Molecular Weight | 410.47 |
Formula | C21H26N6O3 |
CAS No. | 1454808-95-7 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 30 mg/mL (73.09 mM), Sonication is recommended.
You can also refer to dose conversion for different animals. More
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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.
LP-922761 1454808-95-7 Neuroscience AAK1 (AP2 associated kinase 1) LP 922761 LP922761 inhibitor inhibit