Powder: -20°C for 3 years
In solvent: -80°C for 2 years
CB1-IN-1 is a peripherally restricted CB1R antagonist, for CB1R and CB2R with Ki of 0.3 nM and 21 nM,respectively.
Description | CB1-IN-1 is a peripherally restricted CB1R antagonist, for CB1R and CB2R with Ki of 0.3 nM and 21 nM,respectively. |
Targets&IC50 | CB2R:21 nM, CB1R:0.3 nM |
Synonyms | DBPR211, 1-(2,4-二氯苯基)-N-1-哌啶基-4-[[(1-吡咯烷基磺酰基)氨基]甲基]-5-[5-[2-[4-(三氟甲基)苯基]乙炔基]-2-噻吩基]-1H-吡唑-3-甲酰胺 |
Molecular Weight | 751.67 |
Formula | C33H31Cl2F3N6O3S2 |
CAS No. | 1429239-98-4 |
Powder: -20°C for 3 years
In solvent: -80°C for 2 years
DMSO: 10 mM
( < 1 mg/ml refers to the product slightly soluble or insoluble )
You can also refer to dose conversion for different animals. More
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CB1-IN-1 1429239-98-4 G蛋白偶联受体 Cannabinoid Receptor Inhibitor inhibit BPRCB 1184 CB1IN1 BPRCB-1184 BPRCB1184 DBPR211 CB-1-IN-1 CB1 IN 1 inhibitor