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AZD1940

Catalog No. T30252 CAS 881413-29-2

Synonyms: UNII-0J0035E9FT, AZD-1940, AZD 1940

AZD1940 (UNII-0J0035E9FT) is a high affinity CB(1)/CB(2) receptor agonist of the cannabinoid with oral activity. Application in the study of orofacial pain.

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AZD1940, CAS 881413-29-2

Pack Size	Availability	Price/USD
1 mg	In stock	$ 132.00
5 mg	In stock	$ 328.00
10 mg	In stock	$ 563.00
25 mg	In stock	$ 891.00
50 mg	In stock	$ 1,230.00
100 mg	In stock	$ 1,670.00
1 mL * 10 mM (in DMSO)	In stock	$ 363.00

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Purity: 99.43%

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Description	AZD1940 (UNII-0J0035E9FT) is a high affinity CB(1)/CB(2) receptor agonist of the cannabinoid with oral activity. Application in the study of orofacial pain.
In vitro	AZD1940 demonstrates high binding affinity towards the CB1 and CB2 receptors in humans, rats, and mice, exhibiting full agonism at both receptor types across these species[1].
In vivo	After given orally to human, the mean maximum plasma concentration (Cmax) for AZD1940 800 mg was 9.3 nmol/L . The mean concentration over post-dose eight hours for AZD1940 was 236 nmol.h/L[1].

Synonyms	UNII-0J0035E9FT, AZD-1940, AZD 1940
Molecular Weight	413.52
Formula	C20H29F2N3O2S
CAS No.	881413-29-2

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year

Solubility Information

DMSO: 90.0 mg/mL (217.6 mM), Sonication is recommended.

References and Literature

1. Schou M, et al. Radiolabeling of the cannabinoid receptor agonist AZD1940 with carbon-11 and PET microdosing in non-human primate. Nucl Med Biol. 2013 Apr;40(3):410-4. 2. Kalliomäki J, et al. Evaluation of the analgesic efficacy and psychoactive effects of AZD1940, a novel peripherally acting cannabinoid agonist, in human capsaicin-induced pain and hyperalgesia. Clin Exp Pharmacol Physiol. 2013 Mar;40(3):212-8. 3. Grossman S, et al. Cannabis and orofacial pain: a systematic review. Br J Oral Maxillofac Surg. 2022 Jun;60(5):e677-e690.

Related compound libraries

This product is contained In the following compound libraries：

GPCR Compound Library Anti-Cancer Clinical Compound Library Anti-Cancer Drug Library Drug Repurposing Compound Library Clinical Compound Library Neuronal Signaling Compound Library Bioactive Compounds Library Max Bioactive Compound Library

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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.

Keywords

AZD1940 881413-29-2 GPCR/G Protein Cannabinoid Receptor UNII-0J0035E9FT AZD-1940 AZD 1940 inhibitor inhibit

Products are chemical reagents for research use only and are not intended for human use. We do not sell to patients.