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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T60255 | α-Amylase/α-Glucosidase-IN-1 | ||
α-Amylase/α-Glucosidase-IN-1 (compound 33) is an effective inhibitor of α-amylase/α-glucosidase with IC 50 s of 2.01, 2.09 μM for α-amylase and α-glucosidase, respectively. Kinetic studies predict that α-Amylase/α-Glucos... | |||
T61706 | α-Amylase/α-Glucosidase-IN-2 | ||
α-Amylase/α-Glucosidase-IN-2 (compound 5) exhibits strong inhibition activity towards both α-amylase and α-glucosidase enzymes, with IC 50 values of 13.02 μM and 13.09 μM, respectively. This compound shows promise for in... | |||
T79225 | α-Amylase/α-Glucosidase-IN-3 | Glucosidase | |
α-Amylase/α-Glucosidase-IN-3 (Compound 17) serves as a dual inhibitor targeting both α-Amylase and α-Glucosidase, exhibiting IC50 values of 0.70 μM and 1.10 μM, respectively. It is applicable for type-II diabetes mellitu... | |||
T78878 | α-Amylase/α-Glucosidase-IN-5 | Glucosidase | |
α-Amylase/α-Glucosidase-IN-5 (compound 4l) functions as a dual inhibitor, effectively inhibiting both α-glucosidase (Glucosidase) and α-amylase (Amylases) with IC50 values of 5.96 μM and 1.62 μM, respectively, exhibiting... | |||
T80715 | α-Amylase/α-Glucosidase-IN-6 | ||
α-Amylase/α-Glucosidase-IN-6 (compound 5j) serves as a potent dual inhibitor of both α-amylase and α-glucosidase, exhibiting IC50 values of 17.0 µM and 40.1 µM, respectively. It demonstrates anti-hyperglycemic activities... | |||
T79402 | α-Amylase/α-Glucosidase-IN-4 | Glucosidase | |
α-Amylase/α-Glucosidase-IN-4 (compound 5), a dual inhibitor targeting α-amylase (Amylases) and α-glucosidase (Glucosidase), exhibits potent inhibition with IC50 values of 1.10 μM and 0.15 μM respectively. This compound i... | |||
T74255 | HPA-IN-1 | ||
HPA-IN-1 (Compound 1) serves as a potent and selective inhibitor of human pancreatic α-amylase (HPA), demonstrating specificity with IC50 values of 12.0 μM for HPA and 410.4 μM for α-glucosidase [1]. |