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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T79519 | YXG-158 | Androgen Receptor | |
YXG-158 (Compound 23-h), an orally active androgen receptor (AR) degrader and cytochrome P450 17A1 (CYP17A1) inhibitor, exhibits AR degradation with a DC50 of 1.28 μM and CYP17A1 inhibition with an IC50 of 100 nM. It is ... |