3
Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T12679 | (Rac)-VU 6008667 | Others , AChR | |
(Rac)-VU 6008667 is a selective negative allosteric modulator of muscarinic acetylcholine receptor subtype 5 (M5 NAM) with IC50 of 1.8 μM and pIC50 of 5.75, has high CNS penetration. | |||
T13315 | VU 6008667 | Others | |
VU 6008667 is a selective negative allosteric M5 NAM modulator (IC50s: 1.2 μM and 1.6 μM for human M5 and rat M5, respectively). | |||
T12647 | (R)-VU 6008667 | Others | |
(R)-VU 6008667 is devoid of M5 NAM activity (IC50>10 μM). |