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Search Results for " sb-216469 "

2

Compounds

Cat No. Product Name Synonyms Targets
T9762 Upidosin SB-216469,SB 216469,Rec 15-2739,Recordati 15/2739 Adrenergic Receptor
Upidosin (SB-216469) is a potential uroselective α1-adrenoceptor antagonist, α1a subtype Ki=0.34 nM, α1b subtype Ki=3.9 nM, α1d subtype Ki=1.5 nM, α2-adrenoceptor Ki=33.3 nM.
T37794 Rec 15/2615 (hydrochloride)
Rec 15/2615 is an antagonist of α1B-adrenergic receptors (α1B-ARs; Ki = 0.45 nM for the recombinant human receptor).1 It selectively inhibits α1B-ARs over α1A-, α1D-, and α1L-ARs (Kis = 7.59, 10.23, and 49 nM, respective...
TargetMol