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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T6240 | Palbociclib Isethionate | Palbociclib (PD0332991) Isethionate,PD 0332991 isethionate | CDK |
Palbociclib Isethionate (PD 0332991 isethionate) is a selective inhibitor of CDK4/6 (IC50s: 11/16 nM). It exhibits no inhibition against a panel of 36 additional protein kinases. | |||
T1785 | Palbociclib | PD 0332991 | CDK |
Palbociclib (PD 0332991) is a CDK inhibitor that inhibits CDK4 and CDK6 (IC50=11/16 nM) and is orally active. Palbociclib has anti-tumorigenic activity and has investigational potential for use in ER-positive and HER2-ne... | |||
T33865 | Palbociclib-SMCC | PD0332991-SMCC,Palbociclib-SMCC linker,PD 0332991-SMCC,PD-0332991-SMCC | |
Palbociclib-SMCC is a Palbociclib derivative with a SMCC linker. | |||
T6239 | Palbociclib monohydrochloride | PD 0332991 hydrochloride,Palbociclib hydrochloride,Palbociclib (PD-0332991) HCl | CDK |
Palbociclib monohydrochloride (PD 0332991 hydrochloride) is a selective inhibitor of CDK4/6 (IC50s: 11/16 nM). It exhibits no inhibition against a panel of 36 additional protein kinases. |