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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T11338 | Furamidine | DB75,NSC 305831 | Others |
Furamidine is also a selective and cell-permeable protein arginine methyltransferase 1 (PRMT1) inhibitor with an IC50 of 9.4 μM. Furamidine is selective for PRMT1 over PRMT5, PRMT6, and PRMT4 (CARM1) (IC50s of 166 μM, 28... | |||
T27395 | Furamidine dihydrochloride | DB 75, DB75, NSC 305831, WR199385,Furamidine HCl | |
Furamidine is a cell-permeable, selective inhibitor of protein arginine methyltransferase 1 (PRMT1). Furamidine binds to strings of AT base pair sequences in DNA′s minor groove. Furamidine targets the enzyme active site ... |